SCHEMBL17185501

SCHEMBL17185501

COC(=O)c1cc(Oc2ccc(C(=O)OC(C)(C)C)cc2)c(C)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
FPR2 P25090 2/20 0.38
SCN9A Q15858 2/20 0.38
NOTUM Q6P988 1/20 0.38
MET P08581 1/20 0.38
AXL P30530 1/20 0.38
RXRA P19793 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
PDGFRB P09619 1/20 0.37
FGFR1 P11362 1/20 0.37
PDGFRA P16234 1/20 0.37
FLT1 P17948 1/20 0.37
FGFR3 P22607 1/20 0.37
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17185192 0.81 LMNA (0.46) KMT2AHPGDNPSR1LMNATDP1
SCHEMBL31063578 0.80 CA1 (0.42) ALDH1A1HPGDNPSR1KDM4ECA1
SCHEMBL31063581 0.79 TDP1 (0.43) ALDH1A1NPSR1KDM4ECA1CA2
SCHEMBL31455709 0.76 NOTUM (0.38) ALDH1A1HPGDSCN9ANOTUMKDM4E
SCHEMBL24515578 0.76 LMNA (0.45) ALDH1A1HPGDAXLKDM4EPOLB
SCHEMBL24515938 0.74 CYP1A2 (0.44) ALDH1A1KMT2AHPGDKDM4EPOLB
SCHEMBL4466049 0.74 CA12 (0.42) ALDH1A1KMT2AHPGDNPSR1RXRA
SCHEMBL17184697 0.73 KDM4E (0.51) ALDH1A1KMT2AHPGDKDM4EPOLB
SCHEMBL5918245 0.72 HPGD (0.54) ALDH1A1KMT2AHPGDCA1CA2
SCHEMBL3990255 0.72 KDM4E (0.47) ALDH1A1HPGDNOTUMKDM4ECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161011-A1 BENZAMIDE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed