SCHEMBL17185192

SCHEMBL17185192

COC(=O)c1cc(Oc2ccc(Cl)cc2)c(C)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.46
PNLIP P16233 5/20 0.44
TDP1 Q9NUW8 1/20 0.44
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
ABL1 P00519 1/20 0.42
KMT2A Q03164 1/20 0.42
P2RX3 P56373 2/20 0.41
HPGD P15428 1/20 0.41
EPAS1 Q99814 1/20 0.41
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364360 0.83 LMNA (0.43) LMNAPNLIPTDP1CCNCCDK8
SCHEMBL17185349 0.82 HTR2A (0.42) LMNAPNLIPTDP1CCNCCDK8
SCHEMBL17185501 0.81 ALDH1A1 (0.40) LMNATDP1KMT2AHPGDL3MBTL1
SCHEMBL17996051 0.80 P2RX3 (0.55) LMNATDP1ABL1P2RX3SLC6A4
SCHEMBL4449413 0.78 PTGER4 (0.57) LMNAPNLIPTDP1ABL1HPGD
SCHEMBL17184697 0.78 KDM4E (0.51) KMT2AHPGDMAPT
SCHEMBL363951 0.75 GAA (0.46) LMNAABL1KMT2AHPGDNPC1
SCHEMBL1462096 0.74 ABL1 (0.61) LMNAABL1KMT2AHPGDSLC6A4
SCHEMBL5357436 0.74 TDP1 (0.53) LMNAPNLIPTDP1ABL1KMT2A
SCHEMBL19993672 0.74 MAPT (0.42) LMNATDP1HPGDSLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161011-A1 BENZAMIDE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed