SCHEMBL17196427

SCHEMBL17196427

CCc1ncc(C(C)(C)O)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
MAPT P10636 1/20 0.34
MAOB P27338 1/20 0.34
GABRB3 P28472 2/20 0.34
GABRA2 P47869 2/20 0.34
GABRB2 P47870 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
GLA P06280 1/20 0.33
CDC7 O00311 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24424827 0.84 TDP1 (0.41) L3MBTL1TDP1KMT2AMEN1NPSR1
SCHEMBL29585732 0.84 TDP1 (0.41) L3MBTL1TDP1KMT2AMEN1NPSR1
SCHEMBL21419164 0.81 AGBL2 (0.44) MAOBCDC7PLK4CHEK1AURKA
SCHEMBL30861680 0.80 TDP1 (0.58) L3MBTL1TDP1KMT2AMEN1NPSR1
SCHEMBL9290492 0.80 TDP1 (0.58) L3MBTL1TDP1KMT2AMEN1NPSR1
SCHEMBL30861677 0.80 TDP1 (0.58) L3MBTL1TDP1KMT2AMEN1NPSR1
Ammonia Solution, Strong SCHEMBL20298816 0.79 TDP1 (0.56) L3MBTL1TDP1KMT2AMEN1NPSR1
SCHEMBL2415072 0.77 ALDH1A1 (0.42) KMT2AMEN1NPSR1MAOBALDH1A1
SCHEMBL17173641 0.76 ALDH1A1 (0.36) KMT2ACYP2C19HTTRAB9AMAOB
SCHEMBL17177782 0.76 CHRNB2 (0.38) L3MBTL1KMT2AHTTMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015158427-A1 HETEROARYL SUBSTITUTED HETEROCYCLYL SULFONES Grünenthal GmbH (DE) 2015-10-22 WO disclosed