SCHEMBL171978

SCHEMBL171978

Cc1ccc2c(cnn2I)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
CYP2A6 P11509 3/20 0.41
CYP1A2 P05177 2/20 0.41
NR3C1 P04150 2/20 0.40
MAPT P10636 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
POLB P06746 1/20 0.37
KMO O15229 1/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25044243 0.78 NOS1 (0.38) CYP11B2MAPT
SCHEMBL424964 0.78 TRPA1 (0.46) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2
SCHEMBL29769166 0.78 TRPA1 (0.46) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2
SCHEMBL15185701 0.76 SLC22A12 (0.47) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2
SCHEMBL13486145 0.76 NR3C1 (0.61) CYP11B1CYP11B2NR3C1
SCHEMBL16648362 0.76 SLC22A12 (0.43) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2
SCHEMBL29520791 0.76 NR3C1 (0.43) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2
SCHEMBL3657596 0.76 CYP11B1 (0.47) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2
SCHEMBL14765172 0.76 HDAC8 (0.39) CYP11B1CYP11B2CYP2A6MAPTHDAC8
SCHEMBL19772304 0.76 SLC22A12 (0.40) SLC22A12CYP11B1CYP11B2CYP2A6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023107673-A2 CLEAVABLE DISULFIDE LINKERS AND USES THEREOF Singular Genomics Systems, Inc. (US) 2023-06-15 WO disclosed
EP-3892616-A1 AROMATIC RING DERIVATIVE AS IMMUNOREGULATION AND PREPARATION METHOD AND APPLICATION OF AROMATIC RING DERIVATIVE Shanghai Jemincare Pharmaceuticals Co., Ltd. (CN) 2021-10-13 EP disclosed
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed
EP-2426125-A1 1,4 disubstituted 3 cyano pyridone derivatives and their use as positive allosteric modulators of mGluR2 receptors Ortho-McNeil-Janssen Pharmaceuticals, Inc. (US) 2012-03-07 EP disclosed