SCHEMBL172044

SCHEMBL172044

N=Cc1c(Cl)ccc(Cl)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2A6 P11509 1/20 0.32
AHR P35869 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4871529 0.74 ALDH1A1 (0.55) TDP1MEN1ALDH1A1KMT2ACYP2A6
SCHEMBL22681399 0.73 TDP1 (0.60) MAPK1TDP1ALDH1A1
SCHEMBL189622 0.72 ALDH1A1 (0.59) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL14223535 0.72 ALDH1A1 (0.39) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL16958731 0.72 CYP3A4 (0.42) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL5413852 0.72 CYP3A4 (0.36) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL11340423 0.69 ALDH1A1 (0.38) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL11340421 0.69 ALDH1A1 (0.38) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL17146971 0.67 HTR2A (0.36) CYP3A4
SCHEMBL29368277 0.67 CYP3A4 (0.62) CYP3A4MAPK1TDP1ALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066312-B1 USE OF CHLORINE GUANABENZ DERIVATIVES FOR TREATING POLYGLUTAMINE EXPANSION ASSOCIATED DISEASES CENTRE NAT RECH SCIENT (FR) 2012-03-07 EP disclosed