SCHEMBL5413852

SCHEMBL5413852

C[CH]c1c(Cl)ccc(Cl)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2A6 P11509 1/20 0.32
AHR P35869 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2845041 0.80 TNF (0.36) TDP1MEN1ALDH1A1KMT2A
SCHEMBL1547930 0.74 ALDH1A1 (0.55) TDP1MEN1ALDH1A1KMT2ACYP2A6
SCHEMBL172044 0.72 CYP3A4 (0.36) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL189622 0.72 ALDH1A1 (0.59) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL14223535 0.72 ALDH1A1 (0.39) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL16958731 0.72 CYP3A4 (0.42) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL1547628 0.70 CYP3A4 (0.40) CYP3A4MAPK1TDP1CYP2A6AHR
SCHEMBL21030288 0.69 CYP3A4 (0.32) CYP3A4MAPK1ALDH1A1
SCHEMBL6413858 0.67 CYP2A6 (0.54) CYP3A4MAPK1TDP1MEN1ALDH1A1
SCHEMBL29368277 0.67 CYP3A4 (0.62) CYP3A4MAPK1TDP1ALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291730-B2 Pyrimidine compounds and their use SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-11-06 US disclosed
US-20050107609-A1 Pyrimidine compounds and their use SUMITOMO CHEMICAL COMPANY 2005-05-19 US disclosed
US-6838463-B2 Pyrimidine compounds and their use SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2005-01-04 US disclosed
EP-1366026-B1 PYRIMIDINE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2004-12-01 EP disclosed
US-20040077669-A1 Pyrimidine compounds and their use SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-04-22 US disclosed
EP-1366026-A2 PYRIMIDINE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2003-12-03 EP disclosed
WO-2002024663-A2 PYRIMIDINE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050107609-A1 Pyrimidine compounds and their use TYMP, TYMS, UMPS CYP3A4 178/4885MAPK1 2068/4885TDP1 263/4885
US-20040077669-A1 Pyrimidine compounds and their use TYMP, TYMS, DPYD CYP3A4 325/4885MAPK1 1924/4885TDP1 95/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.