SCHEMBL1720696

SCHEMBL1720696

O=C(O)c1ccnc(C(F)(F)F)c1F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASPH Q12797 3/20 0.59
KDM4E B2RXH2 3/20 0.59
KDM8 Q8N371 2/20 0.59
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NAPRT Q6XQN6 2/20 0.43
KDM4A O75164 1/20 0.41
RAB9A P51151 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
HIF1AN Q9NWT6 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC6A9 P48067 1/20 0.41
P2RX7 Q99572 5/20 0.40
DHODH Q02127 1/20 0.39
TAS2R14 Q9NYV8 1/20 0.39
PSMD14 O00487 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29882303 1.00 ASPH (0.59) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL28310940 0.88 KDM4E (0.47) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL28311764 0.87 HTT (0.45) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL18988808 0.86 KDM4E (0.56) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL25342306 0.84 KDM4E (0.58) ASPHKDM4EKDM8NAPRTKDM4A
SCHEMBL1720768 0.84 L3MBTL1 (0.46) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL17509160 0.84 P2RX7 (0.42) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL9928615 0.84 SLC6A9 (0.42) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL2582882 0.80 KDM4E (0.44) ASPHKDM4EKDM8HTTHSD17B10
SCHEMBL29760859 0.80 KDM4E (0.44) ASPHKDM4EKDM8HTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 188 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110950797-A Preparation method of 2-trifluoromethyl-3-fluoro-4-picolinic acid and derivatives thereof 丽水绿氟科技有限公司 2020-04-03 CN claimed
CN-110627714-A Synthetic method of 3-fluoro-2-trifluoromethyl isonicotinic acid 安庆博曼生物技术有限公司 2019-12-31 CN claimed
EP-4682149-A1 POLYMORPH OF JAK TYROSINE KINASE INHIBITOR AND USE THEREOF Prime Gene Therapeutics Co., Ltd. (CN) 2026-01-21 EP disclosed
US-20250346600-A1 TRICYCLIC DERIVATIVES AND RELATED USES MOMA THERAPEUTICS, INC. 2025-11-13 US disclosed
WO-2025233901-A1 ACTIVATORS OF PYRUVATE KINASE ISOFORM M2 AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE BIOHAVEN THERAPEUTICS LTD. (VG) 2025-11-13 WO disclosed
WO-2025054488-A1 TRICYCLIC DERIVATIVES AND RELATED USES MOMA THERAPEUTICS, INC. (US) 2025-03-13 WO disclosed
US-20250034170-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2025-01-30 US disclosed
WO-2024193495-A1 FUMARATE CRYSTAL FORM OF JAK TYROSINE KINASE INHIBITOR, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 北京普祺医药科技股份有限公司 2024-09-26 WO disclosed
WO-2024193496-A1 METHOD FOR PREPARING PYRROLOPYRIMIDINE COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 北京普祺医药科技股份有限公司 2024-09-26 WO disclosed
EP-4415706-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-08-21 EP disclosed
US-12065441-B2 Pyrazolopyrimidine derivative, use thereof and pharmaceutical composition Gengle Therapeutics, Inc. (CN) 2024-08-20 US disclosed
US-20120295884-A1 Complement pathway modulators and uses thereof NOVARTIS AG (CH) 2012-11-22 US disclosed
WO-2012093101-A1 INDOLE COMPOUNDS OR ANALOGUES THEREOF USEFUL FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION (AMD) NOVARTIS AG (CH) 2012-07-12 WO disclosed
US-20120149681-A1 CYCLOBUTYL SUBSTITUTED PYRROLOPYRIDINE AND PYRROLOPYRIMIDINE DERIVATIVES AS JAK INHIBITORS INCYTE CORPORATION 2012-06-14 US disclosed
WO-2012068450-A1 CYCLOBUTYL SUBSTITUTED PYRROLOPYRIDINE AND PYRROLOPYRIMIDINE DERIVATIVES AS JAK INHIBITORS INCYTE CORPORATION (US) 2012-05-24 WO disclosed
EP-2406265-A2 SUBSTITUTED 3-AMINOISOXAZOLOPYRIDINES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2012-01-18 EP disclosed
US-20110224190-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS INCYTE CORPORATION 2011-09-15 US disclosed
WO-2011112662-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS INCYTE CORPORATION (US) 2011-09-15 WO disclosed
WO-2010102778-A2 SUBSTITUTED 3-AMINOISOXAZOLOPYRIDINES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2010-09-16 WO disclosed
US-20100234419-A1 SUBSTITUTED 3-AMINOISOXAZOLOPYRIDINES AS KCNQ2/3 MODULATORS GRUNENTHAL GMBH (DE) 2010-09-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250034170-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF GBA1, GAA, GBA2 ASPH 2393/4885KDM4E 3762/4885KDM8 3760/4885
US-20120295884-A1 Complement pathway modulators and uses thereof C5, C3AR1, C9 ASPH 2393/4885KDM4E 4092/4885KDM8 4026/4885
US-20120149681-A1 CYCLOBUTYL SUBSTITUTED PYRROLOPYRIDINE AND PYRROLOPYRIMIDINE DERIVATIVES AS JAK INHIBITORS JAK1, JAK2, JAK3 ASPH 2421/4885KDM4E 818/4885KDM8 541/4885
US-20100234419-A1 SUBSTITUTED 3-AMINOISOXAZOLOPYRIDINES AS KCNQ2/3 MODULATORS KCNQ1, KCNQ2, KCNQ3 ASPH 4000/4885KDM4E 328/4885KDM8 1561/4885
US-20110224190-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS JAK1, JAK2, JAK3 ASPH 3087/4885KDM4E 248/4885KDM8 972/4885
US-12065441-B2 Pyrazolopyrimidine derivative, use thereof and pharmaceutical composition JAK2, JAK1, JAK3 ASPH 3832/4885KDM4E 2256/4885KDM8 1668/4885
US-20250346600-A1 TRICYCLIC DERIVATIVES AND RELATED USES WRN, RECQL, BLM ASPH 3464/4885KDM4E 3487/4885KDM8 2043/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.