SCHEMBL17209263

SCHEMBL17209263

COc1ccc(CNC(=O)NCCc2cc3ccccc3s2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.54
KMT2A Q03164 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 2/20 0.50
CLK1 P49759 2/20 0.48
PTPN1 P18031 2/20 0.48
NAMPT P43490 1/20 0.48
FPR2 P25090 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
GAA P10253 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HDAC1 Q13547 1/20 0.46
CASP3 P42574 1/20 0.46
POLB P06746 1/20 0.46
GSK3B P49841 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17209265 0.86 EPHX1 (0.49) KMT2AMEN1NAMPTHDAC1POLB
SCHEMBL17202891 0.85 ALDH1A1 (0.57) KMT2AKDM4EALDH1A1NPC1RAB9A
SCHEMBL17209261 0.85 NAMPT (0.53) ALDH1A1NAMPT
SCHEMBL17209262 0.81 TRPV1 (0.47) KMT2AMEN1ALDH1A1EPHX1
SCHEMBL16562237 0.78 EPHX1 (0.74) CASRKMT2AMEN1ALDH1A1NPC1
SCHEMBL17209264 0.77 MAPT (0.50) KMT2AKDM4EMEN1ALDH1A1NAMPT
SCHEMBL1806012 0.77 CYP2A6 (0.50) KMT2AMEN1RAB9ANAMPTHDAC1
SCHEMBL5338788 0.75 KMT2A (0.56) KMT2AKDM4EMEN1ALDH1A1NPC1
SCHEMBL16562080 0.75 NPC1 (0.77) CASRKMT2AKDM4EMEN1ALDH1A1
SCHEMBL12113008 0.74 FPR2 (0.61) CASRKMT2AMEN1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015162216-A1 BIARYL AMIDE OR UREA DERIVATIVES AS TRPV1 LIGANDS UNIVERSITA' DEGLI STUDI DI SIENA (IT) 2015-10-29 WO disclosed