SCHEMBL1721602

SCHEMBL1721602

CNC(=O)C1(C)CC[C@]2(C)CC[C@]3(C)[C@H](CC(=O)[C@@H]4[C@@]5(C)CCCC(C)(C)C5CC[C@]43C)[C@H]2C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.47
TERT O14746 1/20 0.35
NR4A1 P22736 1/20 0.35
HSD11B1 P28845 7/20 0.34
HSD11B2 P80365 6/20 0.34
CYP3A4 P08684 2/20 0.34
TSHR P16473 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTPN2 P17706 1/20 0.32
CYP19A1 P11511 1/20 0.31
CES2 O00748 2/20 0.31
CES1 P23141 2/20 0.31
MAPT P10636 2/20 0.30
MEN1 O00255 1/20 0.30
AKR1B10 O60218 1/20 0.30
LMNA P02545 1/20 0.30
ALOX5 P09917 1/20 0.30
PRKCH P24723 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1721886 0.92 PTPN1 (0.47) PTPN1HSD11B1HSD11B2CYP3A4TSHR
SCHEMBL1721806 0.90 PTPN1 (0.44) PTPN1HSD11B1HSD11B2CYP3A4TSHR
SCHEMBL1721809 0.83 PTPN1 (0.67) PTPN1PTPN2CES2CES1
SCHEMBL418948 0.78 HSD11B1 (0.57) PTPN1HSD11B1HSD11B2CYP3A4TSHR
SCHEMBL420589 0.77 HSD11B1 (0.46) PTPN1HSD11B1HSD11B2CYP3A4TSHR
SCHEMBL418949 0.76 HSD11B1 (0.59) PTPN1HSD11B1HSD11B2CYP3A4TSHR
SCHEMBL421440 0.76 HSD11B1 (0.49) HSD11B1HSD11B2CES2CES1
SCHEMBL421484 0.76 HSD11B1 (0.48) PTPN1HSD11B1HSD11B2CYP3A4TSHR
SCHEMBL418097 0.74 HSD11B1 (0.60) PTPN1HSD11B1HSD11B2CES2CES1
SCHEMBL421285 0.73 HSD11B1 (0.47) HSD11B1HSD11B2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406272-A1 N-HYDROXY C29-AMIDE DERIVATIVES OF OLEANDRANE onepharm Research & Development GmbH (AT) 2012-01-18 EP disclosed