SCHEMBL17220190

SCHEMBL17220190

N=C(NO)c1nc(N)nc(NCc2ccccc2Cl)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HRH4 Q9H3N8 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
ADORA2A P29274 3/20 0.42
ADORA1 P30542 1/20 0.42
MAP4K4 O95819 1/20 0.39
HTR2B P41595 1/20 0.38
GPR68 Q15743 1/20 0.38
TP53 P04637 1/20 0.38
CD38 P28907 1/20 0.38
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17220394 0.85 VNN1 (0.42) ADORA2AADORA1MAP4K4HTR2BGPR68
SCHEMBL14869738 0.82 HRH4 (0.53) HDAC3HDAC1HDAC2HDAC6HRH4
SCHEMBL17220071 0.74 KCNH3 (0.44) HRH4HRH3GPR68HTR7HTR6
SCHEMBL17220381 0.72 APP (0.50) HRH4ADORA2AADORA1GPR68HTR1A
SCHEMBL796783 0.72 LMNA (0.40) HDAC3HDAC1HDAC2HDAC6NPC1
SCHEMBL796546 0.72 NPC1 (0.50) HDAC6TP53ALDH1A1NPC1RAB9A
SCHEMBL14869762 0.72 HRH4 (0.48) HRH4HRH3ADORA2AMAP4K4TP53
SCHEMBL14869876 0.72 HRH4 (0.48) HRH4HRH3ADORA2AMAP4K4HTR2B
SCHEMBL4377934 0.71 HTR2B (0.54) HDAC1ADORA2AHTR2BGPR68HTR1A
SCHEMBL17220209 0.69 HDAC3 (0.48) HDAC3HDAC1HDAC2HDAC6HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616465-B1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2015-11-04 EP disclosed