SCHEMBL17220071

SCHEMBL17220071

N=C(NO)c1nc(N)nc(NCc2ccc(F)cc2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 4/20 0.44
APP P05067 1/20 0.44
GPR68 Q15743 3/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
ADRA1D P25100 1/20 0.40
HTR2C P28335 1/20 0.40
HTR7 P34969 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
HTR6 P50406 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17220381 0.85 APP (0.50) APPGPR68HRH4NPSR1
SCHEMBL29223873 0.81 CA1 (0.60) KCNH3APPGPR68CA1CA2
SCHEMBL17220394 0.79 VNN1 (0.42) GPR68KDM4EMEN1KMT2AVNN1
SCHEMBL17220378 0.74 DHFR (0.43) CA9KDM4EHSD17B10NPSR1
SCHEMBL17220190 0.74 HDAC3 (0.48) GPR68HRH4HRH3HTR7HTR6
SCHEMBL796742 0.71 TP53 (0.47) CA9KDM4EMEN1KMT2AHSD17B10
SCHEMBL17173044 0.70 KCNH3 (0.51) KCNH3APPGPR68CA1CA2
SCHEMBL17220339 0.70 RAB9A (0.45) KDM4EMEN1KMT2AATMHSD17B10
SCHEMBL17220072 0.69 DHFR (0.31) APP
SCHEMBL17220062 0.69 CGAS (0.45) APPCA1CA2CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616465-B1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2015-11-04 EP disclosed