SCHEMBL1724832

SCHEMBL1724832

CCOC(=O)c1csc(-c2ccnc(N)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.53
DBF4 Q9UBU7 3/20 0.53
CDK5 Q00535 1/20 0.52
CDK5R1 Q15078 1/20 0.52
ALDH1A1 P00352 7/20 0.45
HSD17B10 Q99714 4/20 0.45
HPGD P15428 3/20 0.45
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAOA P21397 1/20 0.44
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
CHEK2 O96017 1/20 0.42
MAPT P10636 5/20 0.42
RAB9A P51151 5/20 0.42
MEN1 O00255 4/20 0.42
NPC1 O15118 4/20 0.42
KMT2A Q03164 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL939732 0.83 ALDH1A1 (0.52) CDC7DBF4CDK5CDK5R1ALDH1A1
SCHEMBL256755 0.80 GABRP (0.56) CDC7DBF4LMNACYP1A2CYP3A4
SCHEMBL16065124 0.80 GSK3B (0.37) CDC7DBF4CDK5CDK5R1ALDH1A1
SCHEMBL938199 0.79 HPGD (0.55) ALDH1A1HSD17B10HPGDLMNAMAPT
Hydrochloric Acid SCHEMBL5591077 0.79 JMJD6 (0.55) CDC7DBF4LMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL6740832 0.79 JMJD6 (0.55) CDC7DBF4LMNACYP1A2CYP3A4
SCHEMBL1724052 0.79 GABRP (0.59) CDC7DBF4ALDH1A1MKNK1MKNK2
SCHEMBL5237356 0.77 MAPT (0.56) ALDH1A1HPGDMAPTRAB9AMEN1
SCHEMBL9454728 0.77 HSD17B10 (0.53) CDC7DBF4ALDH1A1HSD17B10HPGD
SCHEMBL31704904 0.77 CYP2C9 (0.47) CDC7DBF4ALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403857-A1 THIENOPYRIMIDINE AS CDC7 KINASE INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2012-01-11 EP disclosed
WO-2010101302-A1 THIENOPYRIMIDINE AS CDC7 KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-10 WO disclosed