SCHEMBL172491

SCHEMBL172491

O=C(O)c1c(-c2ccc(F)cc2)nn2ccc3c(c12)CCO3

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.52
MTNR1B P49286 10/20 0.52
KMT2A Q03164 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRNA3 P32297 1/20 0.34
HTR3A P46098 1/20 0.34
KCNH2 Q12809 1/20 0.34
UGCG Q16739 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPK14 Q16539 2/20 0.33
MAPK1 P28482 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
EED O75530 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL172381 0.90 MTNR1B (0.62) MTNR1AMTNR1BKMT2ATSHREED
SCHEMBL128044 0.87 MTNR1A (0.51) MTNR1AMTNR1BKMT2AALDH1A1LMNA
SCHEMBL124654 0.81 MTNR1A (0.53) MTNR1AMTNR1BMAPK14EED
SCHEMBL172456 0.78 MTNR1B (0.60) MTNR1AMTNR1BKMT2AL3MBTL1
SCHEMBL125589 0.78 MTNR1A (0.63) MTNR1AMTNR1BKMT2AALDH1A1LMNA
SCHEMBL126984 0.77 MTNR1B (0.82) MTNR1AMTNR1B
SCHEMBL172421 0.77 MTNR1A (0.54) MTNR1AMTNR1BMAPK14EED
Hydrochloric Acid SCHEMBL130262 0.76 MTNR1A (0.53) MTNR1AMTNR1BMAPK14EED
SCHEMBL124932 0.76 MTNR1A (0.48) MTNR1AMTNR1BMAPK14EED
SCHEMBL126117 0.76 MTNR1B (0.71) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100895-B1 TRICYCLIC COMPOUND AND MEDICAL USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2012-03-07 EP disclosed