SCHEMBL17255757

SCHEMBL17255757

COc1cccc(NCCCN2CCN(C)CC2)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.49
CYP2D6 P10635 2/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
KMT2A Q03164 1/20 0.49
TSHR P16473 2/20 0.47
PGK1 P00558 1/20 0.45
POLB P06746 2/20 0.45
HPGD P15428 1/20 0.45
UBE2N P61088 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HTR1A P08908 4/20 0.44
ADRA1A P35348 4/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1B P35368 2/20 0.44
DRD2 P14416 3/20 0.43
CYP3A4 P08684 2/20 0.43
ADRA2A P08913 2/20 0.43
ADRA2B P18089 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072190 0.92 L3MBTL1 (0.51) L3MBTL1CYP2D6MEN1ALDH1A1CYP1A2
SCHEMBL12433870 0.77 CHRM2 (0.51) L3MBTL1ALDH1A1CYP1A2TSHRPOLB
SCHEMBL11808662 0.74 CHRM2 (0.46) L3MBTL1ALDH1A1KMT2ATSHRPOLB
SCHEMBL6402270 0.73 KMT2A (0.50) KMT2AHTR1ADRD2ADRA2CHTR2A
SCHEMBL27982786 0.72 TSHR (0.55) L3MBTL1ALDH1A1TSHRPOLBHPGD
Hydrochloric Acid SCHEMBL11676693 0.71 DRD2 (0.60) ALDH1A1KMT2ATSHRHTR1AADRA1A
Hydrochloric Acid SCHEMBL9129540 0.71 SLC29A1 (0.55) CYP2D6MEN1KMT2ATSHRPGK1
SCHEMBL10831073 0.70 KMT2A (0.47) KMT2ATSHRHPGDNPSR1HTR2A
SCHEMBL24277324 0.70 CHRM2 (0.48) L3MBTL1MEN1ALDH1A1KMT2ATSHR
SCHEMBL24277459 0.70 CHRM2 (0.48) L3MBTL1MEN1ALDH1A1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029543-B1 SUBSTITUTED 3-CYANOPYRIDINES AS PROTEIN KINASE INHIBITORS WYETH LLC (US) 2015-11-18 EP disclosed