SCHEMBL1727464

SCHEMBL1727464

CC(C)Cc1cccc(N2CCC(CCNC(=O)O)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.42
CHRM4 P08173 7/20 0.42
FFAR4 Q5NUL3 1/20 0.40
TRPV3 Q8NET8 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
ACACB O00763 1/20 0.39
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
TGM2 P21980 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1729627 0.86 CHRM4 (0.43) HRH3CHRM4CHRM2CHRM1ACACB
SCHEMBL3269876 0.84 HRH3 (0.40) HRH3CHRM4TRPV3ACACBTGM2
SCHEMBL1728425 0.84 HTR1A (0.51) CHRM4ACACBCKS1BSKP1SKP2
SCHEMBL240061 0.83 HRH3 (0.39) HRH3CHRM4TRPV3ACACBCKS1B
SCHEMBL1728737 0.83 HSD11B1 (0.49) CHRM4CHRM2
SCHEMBL1729311 0.80 HTR1A (0.46) CHRM4FFAR4CHRM2ACACB
SCHEMBL5777613 0.80 HRH3 (0.44) HRH3FFAR4TRPV3ACACB
SCHEMBL14797306 0.79 HSD11B1 (0.44) CHRM4FFAR4ACACBCKS1BSKP1
SCHEMBL1728924 0.79 CNR1 (0.47) CHRM4CKS1BSKP1SKP2TGM2
SCHEMBL1728880 0.78 CHRM4 (0.49) CHRM4CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP claimed
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP disclosed
CN-1812980-B Piperidinyl-and piperazinyl-alkylcarbamate derivatives, their preparation and their use as pharmaceuticals SANOFI AVENTIS 2011-04-06 CN disclosed
CN-101712660-A Piperidinyl-and piperazinyl-alkylcarbamate derivatives, their preparation and their therapeutic use SANOFI AVENTIS 2010-05-26 CN disclosed
CN-1812980-A Piperidinyl-and piperazinyl-alkylcarbamate derivatives, their preparation and their therapeutic use SANOFI AVENTIS (FR) 2006-08-02 CN disclosed
EP-1633735-A1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS Sanofi-Aventis (FR) 2006-03-15 EP disclosed
WO-2004099176-A1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI-AVENTIS (FR) 2004-11-18 WO disclosed