SCHEMBL1728322

SCHEMBL1728322

CCN(C(=O)O)c1cc2c(F)ccc(C)c2nc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
CYP3A4 P08684 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK14 Q16539 2/20 0.34
MAPT P10636 2/20 0.33
CRHR1 P34998 1/20 0.33
TSHR P16473 1/20 0.33
TSPO P30536 1/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
PKM P14618 1/20 0.32
CD38 P28907 1/20 0.32
MAPK1 P28482 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5138 0.75 MAPT (0.32) NPSR1MAPTTSPOKDM4ETP53
SCHEMBL895206 0.72 ALDH1A1 (0.47) ALDH1A1CYP3A4MEN1KMT2AL3MBTL1
SCHEMBL8613 0.72 TP53 (0.43) ALDH1A1CYP3A4NPSR1CYP1A2CYP2D6
SCHEMBL845050 0.71 MAPT (0.37) ALDH1A1CYP3A4MAPK14MAPTTSHR
SCHEMBL1728325 0.71 ALDH1A1 (0.41) ALDH1A1CYP3A4NPSR1CYP1A2CYP2D6
SCHEMBL1883808 0.71 ALDH1A1 (0.41) ALDH1A1CYP3A4NPSR1CYP1A2CYP2D6
SCHEMBL714757 0.69 L3MBTL1 (0.36) ALDH1A1MEN1KMT2AL3MBTL1KDM4E
SCHEMBL1725922 0.68 MAPT (0.51) ALDH1A1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL6976100 0.64 CYP3A4 (0.58) ALDH1A1CYP3A4NPSR1CYP1A2CYP2D6
SCHEMBL10965817 0.64 MEN1 (0.42) ALDH1A1CYP3A4NPSR1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403847-A1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB Pharma, S.A. (BE) 2012-01-11 EP disclosed
WO-2010100405-A1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-09-10 WO disclosed