SCHEMBL17294172

SCHEMBL17294172

CS(=O)(=O)c1ccc(CC2(NO)C(=O)NC(=O)NC2=O)cc1.O=C1NC(=O)C(Cc2ccc3c(c2)OCO3)(NO)C(=O)N1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
PTGS2 P35354 4/20 0.42
PDE5A O76074 1/20 0.42
PTGS1 P23219 2/20 0.42
HTT P42858 2/20 0.41
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
EDNRB P24530 1/20 0.40
EDNRA P25101 1/20 0.40
MEN1 O00255 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PTPN7 P35236 1/20 0.39
DUSP3 P51452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17294177 0.89 HDAC1 (0.46) SMN1; SMN2KMT2AALDH1A1MEN1
SCHEMBL17294147 0.85 MMP2 (0.49) PTGS2
SCHEMBL10576223 0.68 ALDH1A1 (0.46) SMN1; SMN2HTTKMT2AALDH1A1HSD17B10
SCHEMBL4560949 0.68 ALDH1A1 (0.46) SMN1; SMN2HTTKMT2AALDH1A1HSD17B10
SCHEMBL2893747 0.68 ALDH1A1 (0.46) SMN1; SMN2HTTKMT2AALDH1A1HSD17B10
SCHEMBL17294164 0.68 MMP2 (0.43) ALDH1A1POLBHSD17B10
SCHEMBL10073203 0.67 PTGS2 (0.64) PTGS2PDE5APTGS1KMT2AALDH1A1
SCHEMBL7234080 0.65 HDAC1 (0.49) SMN1; SMN2KMT2AALDH1A1MEN1HSD17B10
SCHEMBL7113133 0.65 KMT2A (0.59) SMN1; SMN2KMT2AALDH1A1MEN1HSD17B10
SCHEMBL5749606 0.65 TAAR1 (0.54) SMN1; SMN2KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3148983-A1 N-HYDROXYLAMINO-BARBITURIC ACID DERIVATIVES AS NITROXYL DONORS The Johns Hopkins University (US) 2017-04-05 EP claimed
WO-2015183838-A1 N-HYDROXYLAMINO-BARBITURIC ACID DERIVATIVES AS NITROXYL DONORS THE JOHNS HOPKINS UNIVERSITY (US) 2015-12-03 WO claimed