SCHEMBL172976

SCHEMBL172976

CC[C@H]1CN(Cc2cccc(-c3cccc(C(=O)N[C@H](CC(C)C)CN(C)C)c3)c2)O[C@H]1CO

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.37
UTS2R Q9UKP6 11/20 0.36
CHRM3 P20309 4/20 0.35
CTSB P07858 2/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
CTSL P07711 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL172688 0.90 UTS2R (0.37) HDAC4UTS2RCHRM3CTSBDRD2
SCHEMBL172828 0.85 CTSL (0.34) HDAC4UTS2RTAS1R3TAS1R1CTSL
SCHEMBL13061119 0.79 HDAC4 (0.45) HDAC4UTS2RCTSBTAS1R3TAS1R1
SCHEMBL13060853 0.79 HDAC4 (0.45) HDAC4UTS2RCTSBTAS1R3TAS1R1
SCHEMBL13005434 0.77 HDAC4 (0.45) HDAC4UTS2RCTSBCTSLCTSS
SCHEMBL13005436 0.77 HDAC4 (0.45) HDAC4UTS2RCTSBCTSLCTSS
SCHEMBL172903 0.76 HDAC4 (0.34) HDAC4UTS2RTAS1R3TAS1R1CTSL
SCHEMBL172990 0.72 CTSL (0.33) UTS2RCTSLCTSSCTSK
SCHEMBL13060678 0.71 UTS2R (0.50) UTS2R
SCHEMBL13005956 0.71 TDP1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768966-B1 COUMPOUNDS AND METHODS FOR INHIBITING THE INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS INFINITY DISCOVERY INC (US) 2012-03-07 EP disclosed