SCHEMBL172828

SCHEMBL172828

CC[C@H]1CN(Cc2cccc(-c3cccc(C(=O)N[C@H](CC(C)C)CN(C)C)c3)c2OC)O[C@H]1CO

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.34
CTSS P25774 4/20 0.34
CTSK P43235 3/20 0.34
HDAC4 P56524 1/20 0.34
UTS2R Q9UKP6 6/20 0.33
TAS1R3 Q7RTX0 3/20 0.33
TAS1R1 Q7RTX1 3/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL172903 0.91 HDAC4 (0.34) CTSLCTSSCTSKHDAC4UTS2R
SCHEMBL172990 0.87 CTSL (0.33) CTSLCTSSCTSKUTS2RROCK2
SCHEMBL172976 0.85 HDAC4 (0.37) CTSLCTSSCTSKHDAC4UTS2R
SCHEMBL13060890 0.82 CTSL (0.41) CTSLCTSSCTSKHDAC4UTS2R
SCHEMBL13060892 0.82 CTSL (0.41) CTSLCTSSCTSKHDAC4UTS2R
SCHEMBL13005481 0.80 CTSL (0.41) CTSLCTSSCTSKHDAC4UTS2R
SCHEMBL13005472 0.80 CTSL (0.41) CTSLCTSSCTSKHDAC4UTS2R
SCHEMBL172688 0.75 UTS2R (0.37) HDAC4UTS2R
SCHEMBL13060891 0.75 TAS1R3 (0.44) CTSLCTSSCTSKHDAC4TAS1R3
SCHEMBL13006806 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768966-B1 COUMPOUNDS AND METHODS FOR INHIBITING THE INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS INFINITY DISCOVERY INC (US) 2012-03-07 EP disclosed