SCHEMBL172990

SCHEMBL172990

CC[C@H]1CN(Cc2cccc(-c3cccc(C(=O)N[C@H](CN(C)C)C4CCCCC4)c3)c2OC)O[C@H]1CO

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.33
CTSS P25774 3/20 0.33
UTS2R Q9UKP6 3/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSK P43235 1/20 0.32
CD274 Q9NZQ7 2/20 0.32
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
PDCD1 Q15116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL172828 0.87 CTSL (0.34) CTSLCTSSUTS2RCTSKROCK2
SCHEMBL13060641 0.84 MEN1 (0.41) CTSLCTSSMEN1ALDH1A1MAPK1
SCHEMBL13005623 0.81 BRD4 (0.39) CTSLCTSSMEN1ALDH1A1MAPK1
SCHEMBL172903 0.79 HDAC4 (0.34) CTSLCTSSUTS2RCTSKROCK2
SCHEMBL12269509 0.74 TDP1 (0.32)
SCHEMBL172786 0.74 TDP1 (0.31)
SCHEMBL14186271 0.74 TDP1 (0.31)
SCHEMBL10209001 0.74 TDP1 (0.31)
SCHEMBL172976 0.72 HDAC4 (0.37) CTSLCTSSUTS2RCTSK
SCHEMBL13060644 0.72 CTSS (0.44) CTSLCTSSMEN1KMT2ACTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768966-B1 COUMPOUNDS AND METHODS FOR INHIBITING THE INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS INFINITY DISCOVERY INC (US) 2012-03-07 EP disclosed