SCHEMBL1729975

SCHEMBL1729975

Nc1cccc(F)c1S.Nc1cccc(F)c1S.[Zn]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
CYP3A4 P08684 4/20 0.38
TSHR P16473 3/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
PIK3CA P42336 1/20 0.36
KEAP1 Q14145 1/20 0.32
CD44 P16070 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27543087 1.00 ALDH1A1 (0.38) ALDH1A1CYP3A4TSHRHPGDHSD17B10
SCHEMBL5619974 0.97
SCHEMBL27518041 0.95 ALDH1A1 (0.38) ALDH1A1CYP3A4TSHRHPGDHSD17B10
SCHEMBL27501043 0.95 ALDH1A1 (0.38) ALDH1A1CYP3A4TSHRHPGDHSD17B10
SCHEMBL1817953 0.81 CES2 (0.39) CES2CES1TAAR1
SCHEMBL457725 0.78
SCHEMBL23855444 0.78
SCHEMBL1815421 0.75 CES2 (0.39) CES2CES1TAAR1
SCHEMBL59477 0.70
SCHEMBL601969 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440970-B1 Benzenesulfonic acid salt of 1-(6-halogeno-2-benzothiazolyl)ethylamine IHARA CHEMICAL IND CO (JP) 2011-11-30 EP disclosed
EP-1026163-B1 PROCESS FOR PRODUCING SUBSTITUTED ALKYLAMINES OR SALTS THEREOF IHARA CHEMICAL IND CO (JP) 2006-03-22 EP disclosed
EP-1440970-A1 Process for producing substituted alkylamines or salts thereof IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2004-07-28 EP disclosed
US-6197969-B1 REACTING METAL SALT OF 2-AMINOTHIOPHENOL WITH AN AMINO ACID-N-CARBOXYLIC ANHYDRIDE; CYCLIZATION IN ACID IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2001-03-06 US disclosed
EP-1026163-A1 PROCESS FOR PRODUCING SUBSTITUTED ALKYLAMINES OR SALTS THEREOF IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2000-08-09 EP disclosed