SCHEMBL1733451

SCHEMBL1733451

COc1ccccc1-c1cc(C(N)=O)nc(S(C)(=O)=O)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.61
LMNA P02545 4/20 0.61
NPSR1 Q6W5P4 4/20 0.61
KDM4E B2RXH2 2/20 0.61
HTT P42858 2/20 0.61
MITF O75030 1/20 0.61
STAT3 P40763 1/20 0.61
CHRNA7 P36544 1/20 0.52
KMT2A Q03164 2/20 0.46
SDHB P21912 2/20 0.46
ADORA3 P0DMS8 4/20 0.45
HSP90AA1 P07900 2/20 0.45
ADORA1 P30542 4/20 0.44
ADORA2A P29274 2/20 0.44
HSP90AB1 P08238 1/20 0.44
IKBKB O14920 1/20 0.43
ALDH1A1 P00352 1/20 0.42
TP53 P04637 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HSD17B10 Q99714 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734115 0.86 NPSR1 (0.44) HPGDLMNANPSR1KDM4EHTT
SCHEMBL2816888 0.82 HSP90AA1 (0.52) HPGDLMNANPSR1KDM4EHTT
SCHEMBL1734114 0.79 BPTF (0.57) HPGDLMNANPSR1KDM4EHTT
SCHEMBL1733692 0.79 ADORA3 (0.49) HPGDLMNANPSR1KDM4EHTT
SCHEMBL1734398 0.79 CHRNA7 (0.49) HPGDKDM4ECHRNA7KMT2AADORA3
SCHEMBL1733437 0.77 ADORA3 (0.44) HPGDLMNANPSR1KDM4EHTT
SCHEMBL19805677 0.76 NPSR1 (1.00) HPGDLMNANPSR1KDM4EHTT
SCHEMBL1734511 0.76 KDM4E (0.66) HPGDKDM4ECHRNA7ADORA3HSP90AA1
SCHEMBL1734400 0.74 LMNA (0.45) HPGDLMNANPSR1KDM4EHTT
SCHEMBL30755408 0.74 ALDH1A1 (0.61) HPGDLMNAKDM4EHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8822451-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-09-02 US disclosed
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP disclosed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO disclosed
EP-1891018-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals, Inc. (US) 2008-02-27 EP disclosed
US-20070105833-A1 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED 2007-05-10 US disclosed
WO-2006127588-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070105833-A1 Modulators of ATP-binding cassette transporters ABCC4, CFTR, ABCC2 HPGD 1462/4885LMNA 3617/4885NPSR1 3866/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.