SCHEMBL17339767

SCHEMBL17339767

COc1ccc(CCCNCCOC(c2ccccc2)c2ccc(C)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.67
DRD2 P14416 4/20 0.56
DRD4 P21917 4/20 0.56
DRD3 P35462 4/20 0.56
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
SLC6A3 Q01959 1/20 0.54
HTT P42858 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNA3 P22001 1/20 0.47
HTR1A P08908 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17340063 0.93 SLC6A2 (0.56) SIGMAR1SLC6A2SLC6A4SLC6A3HTT
SCHEMBL17753539 0.93 SIGMAR1 (0.77) SIGMAR1DRD2DRD4DRD3SLC6A2
SCHEMBL8273969 0.90 SIGMAR1 (0.65) SIGMAR1DRD2DRD4DRD3SLC6A2
SCHEMBL17340068 0.84 DRD2 (0.56) SIGMAR1DRD2DRD4DRD3HTT
SCHEMBL17339768 0.84 TP53 (0.54) SIGMAR1HTTMEN1KMT2AHTR1A
SCHEMBL8273974 0.82 SLC6A2 (0.55) SIGMAR1SLC6A2SLC6A4SLC6A3HTT
SCHEMBL17340067 0.81 KCNH2 (0.58) SIGMAR1DRD2DRD4DRD3HTT
SCHEMBL17340053 0.79 SIGMAR1 (0.64) SIGMAR1DRD2DRD4DRD3HTT
SCHEMBL17339771 0.79 CCR3 (0.53) SIGMAR1DRD2DRD4DRD3MEN1
SCHEMBL8099595 0.78 SIGMAR1 (0.68) SIGMAR1DRD2DRD4DRD3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9212127-B2 T type calcium channel inhibitors UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2015-12-15 US disclosed
US-9212127-B2 T type calcium channel inhibitors UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2015-12-15 US disclosed