SCHEMBL173434

SCHEMBL173434

CCOC(=O)c1cnn(CC)c1N

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.68
LMNA P02545 2/20 0.68
ALDH1A1 P00352 6/20 0.62
RAB9A P51151 4/20 0.61
KDM4E B2RXH2 3/20 0.61
HPGD P15428 3/20 0.59
TSHR P16473 3/20 0.58
KMT2A Q03164 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
MEN1 O00255 1/20 0.58
TP53 P04637 1/20 0.54
HTT P42858 2/20 0.53
MAPT P10636 2/20 0.52
ALOX15 P16050 1/20 0.52
HSD17B10 Q99714 1/20 0.52
POLB P06746 1/20 0.50
RECQL P46063 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24452557 0.88 NPC1 (0.65) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL31715213 0.86 NPC1 (0.64) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL7105351 0.86 NPC1 (0.64) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL31352277 0.85 NPC1 (0.62) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL31352167 0.85 NPC1 (0.62) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL1407148 0.84 NPC1 (0.61) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL4242279 0.84 NPC1 (0.61) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL4248164 0.84 NPC1 (0.61) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL17292790 0.84 NPC1 (0.61) NPC1LMNAALDH1A1RAB9AKDM4E
SCHEMBL31715204 0.84 NPC1 (0.61) NPC1LMNAALDH1A1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4737449-A1 P53-Y220C SELECTIVE SMALL-MOLECULAR REACTIVATOR COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF Changchun Genescience Pharmaceutical Co., Ltd. (CN) 2026-05-06 EP disclosed
US-12384764-B2 Pharmaceutical compounds PFIZER INC. (US) 2025-08-12 US disclosed
CN-114787155-B Pharmaceutical compounds 辉瑞公司 2025-02-28 CN disclosed
WO-2025002177-A1 P53-Y220C SELECTIVE SMALL-MOLECULAR REACTIVATOR COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF 长春金赛药业有限责任公司 2025-01-02 WO disclosed
US-20220380349-A1 PHARMACEUTICAL COMPOUNDS PFIZER INC. 2022-12-01 US disclosed
CN-114787155-A Pharmaceutical compounds 瑞威有限公司 2022-07-22 CN disclosed
EP-3324977-B1 BENZODIAZEPINE DERIVATIVES AS RSV INHIBITORS ENANTA PHARM INC (US) 2022-07-13 EP disclosed
WO-2021084280-A1 PHARMACEUTICAL COMPOUNDS ReViral Limited (GB) 2021-05-06 WO disclosed
US-10881666-B2 Combination pharmaceutical agents as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2021-01-05 US disclosed
US-10865215-B2 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2020-12-15 US disclosed
EP-2264037-A1 Vasopressin v1a antagonists Vantia Limited (GB) 2010-12-22 EP disclosed
EP-2264037-A1 Vasopressin v1a antagonists Vantia Limited (GB) 2010-12-22 EP disclosed
EP-2256119-A1 Vasopressin V1a antagonists Vantia Limited (GB) 2010-12-01 EP disclosed
EP-2256119-A1 Vasopressin V1a antagonists Vantia Limited (GB) 2010-12-01 EP disclosed
US-20090029965-A1 Vasopressin V1a Antagonists FERRING B.V. (NL) 2009-01-29 US disclosed
US-20090029965-A1 Vasopressin V1a Antagonists FERRING B.V. (NL) 2009-01-29 US disclosed
US-20090029965-A1 Vasopressin V1a Antagonists FERRING B.V. (NL) 2009-01-29 US disclosed
EP-1781661-A2 VASOPRESSIN V1A ANTAGONISTS Ferring B.V. (NL) 2007-05-09 EP disclosed
WO-2006021213-A2 VASOPRESSIN V1A ANTAGONISTS FERRING B.V. (NL) 2006-03-02 WO disclosed
WO-2006021213-A2 VASOPRESSIN V1A ANTAGONISTS FERRING B.V. (NL) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10865215-B2 Benzodiazepine derivatives as RSV inhibitors GABRA5, GABRA1, GABBR2 NPC1 224/4885LMNA 2153/4885ALDH1A1 621/4885
US-10881666-B2 Combination pharmaceutical agents as RSV inhibitors SERPINB1, FURIN, HIF1AN NPC1 480/4885LMNA 2715/4885ALDH1A1 3562/4885
US-12384764-B2 Pharmaceutical compounds CNR1, HRH4, GABRA1 NPC1 369/4885LMNA 2103/4885ALDH1A1 2411/4885
US-20090029965-A1 Vasopressin V1a Antagonists AVPR1A, AVPR2, AVPR1B NPC1 4072/4885LMNA 2881/4885ALDH1A1 902/4885
US-20220380349-A1 PHARMACEUTICAL COMPOUNDS CNR1, HRH4, GABRA1 NPC1 427/4885LMNA 2197/4885ALDH1A1 2508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.