SCHEMBL17366181

SCHEMBL17366181

N#Cc1ccc(CN2C(=O)c3c(Cl)cccc3C2c2ccc(Cl)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 12/20 0.51
TP53 P04637 3/20 0.45
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CA12 O43570 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CYP19A1 P11511 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17366150 0.83 MDM2 (0.55) MDM2TP53CYP11B1CYP11B2CA12
SCHEMBL17366161 0.83 MDM2 (0.51) MDM2TP53CA12CA2CA9
SCHEMBL30121977 0.72 MDM2 (0.64) MDM2TP53CA12CA9
SCHEMBL17366176 0.70 MDM2 (0.53) MDM2TP53
SCHEMBL21829964 0.68 P2RX3 (0.41) MDM2TP53CYP11B1CYP11B2
SCHEMBL2463170 0.68 MDM2 (1.00) MDM2TP53
SCHEMBL17366169 0.67 MDM2 (0.58) MDM2TP53CA12CA9
SCHEMBL17366151 0.67 MDM2 (0.58) MDM2TP53
SCHEMBL17366174 0.67 MDM2 (0.58) MDM2TP53
SCHEMBL17366167 0.67 MDM2 (0.48) MDM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2960233-B1 NEW THERAPEUTIC AGENTS CANCER RESEARCH TECH LTD (GB) 2019-10-30 EP disclosed
EP-2960233-A1 NEW THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2015-12-30 EP disclosed