SCHEMBL17396387

SCHEMBL17396387

COc1cccc(CN2CC(=O)N(C)Cc3cnc(Cl)nc32)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 6/20 0.43
TNIK Q9UKE5 2/20 0.43
CLPP Q16740 1/20 0.42
CYP3A4 P08684 6/20 0.42
USP2 O75604 5/20 0.42
CYP1A2 P05177 4/20 0.42
CYP2D6 P10635 3/20 0.42
CYP2C9 P11712 3/20 0.42
HSD17B10 Q99714 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
CMA1 P23946 1/20 0.42
CYP2C19 P33261 4/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17396511 0.86 ALDH1A1 (0.40) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL17396567 0.74 TTK (0.54)
SCHEMBL17396447 0.73 ALDH1A1 (0.37) MEN1KMT2AALDH1A1TNIKCLPP
SCHEMBL17396413 0.73 HCRTR1 (0.39) CLPPLMNA
SCHEMBL28734416 0.72 HDAC6 (0.40) MEN1KMT2AALDH1A1CLPPCMA1
SCHEMBL29721827 0.72 HDAC6 (0.40) MEN1KMT2AALDH1A1CLPPCMA1
SCHEMBL17396481 0.71 USP1 (0.41)
SCHEMBL28637841 0.69 FGFR4 (0.48) MAPT
SCHEMBL16071565 0.69 FGFR4 (0.55)
SCHEMBL27810553 0.68 GAA (0.47) KMT2AALDH1A1CLPPALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016001077-A1 COMPOUNDS INHIBITING THE ENZYME MONOPOLAR SPINDLE 1 KINASE,PHARMACEUTICAL COMPOSITIONS AND USES THEREOF IEO - ISTITUTO EUROPEO DI ONCOLOGIA S.R.L. (IT) 2016-01-07 WO disclosed