SCHEMBL174086

SCHEMBL174086

CC1CCC(c2ncc(-c3ccc(Nc4ccc(C(C)(C)C)cc4)cc3)o2)CC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 3/20 0.46
TP53 P04637 6/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 2/20 0.44
NOD2 Q9HC29 1/20 0.44
MAPT P10636 6/20 0.44
PAX8 Q06710 1/20 0.44
LMNA P02545 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL174087 0.86 KMT2A (0.53) KMT2ATP53NPC1RAB9AMAPT
SCHEMBL174631 0.85 KMT2A (0.50) KMT2ACA12CA1CA2CA9
SCHEMBL164685 0.76 KMT2A (0.52) KMT2ATP53NPC1MAPTLMNA
SCHEMBL164651 0.74 KMT2A (0.50) KMT2ATP53NPC1RAB9ANOD2
SCHEMBL173719 0.74 DGAT1 (0.40) LMNA
SCHEMBL12498922 0.69 CA12 (0.61) KMT2ACA12CA1CA2CA9
SCHEMBL19399052 0.68 NPC1 (0.62) KMT2ACA12CA1CA2CA9
SCHEMBL19366465 0.66 HDAC4 (0.65) KMT2ACA12CA1CA2CA9
SCHEMBL12499755 0.66 CA12 (0.57) KMT2ACA12CA1CA2CA9
SCHEMBL2957181 0.66 KIF11 (0.57) KMT2ANPC1RAB9AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed