SCHEMBL17416645

SCHEMBL17416645

CCc1c(OC)cccc1C(=O)N(NC(C)(C)C)C(=O)c1cccc(C)n1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
P2RX7 Q99572 1/20 0.37
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
ALDH1A1 P00352 1/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
KDM4E B2RXH2 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
GAA P10253 1/20 0.34
ABCB1 P08183 1/20 0.34
ADORA2A P29274 1/20 0.34
CSF1R P07333 1/20 0.34
GRM5 P41594 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17416629 0.84 CTSD (0.43) HPGDKDM4ERXFP1LMNA
SCHEMBL9101240 0.82 MAPK1 (0.43) KMT2AMEN1KDM4ECD274LMNA
SCHEMBL17025773 0.82 POLB (0.43) KMT2AMEN1POLBTHRBKDM4E
SCHEMBL2482845 0.81 ABCB1 (0.51) ABCB1
SCHEMBL5053826 0.80 ABCB1 (0.51) KMT2AP2RX7ABCB1
SCHEMBL9100311 0.80 RAB9A (0.43) GAAABCB1MAPTLMNA
SCHEMBL18091874 0.79 MAPT (0.43) KMT2AMEN1POLBHPGDKDM4E
SCHEMBL9102868 0.79 TSHR (0.40) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL27356523 0.78 KDM4E (0.39) KMT2AMEN1ALDH1A1HPGDKDM4E
SCHEMBL18091865 0.78 NPC1 (0.48) KMT2AMEN1ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463269-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-09-28 EP disclosed
EP-2460786-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-01-13 EP disclosed