SCHEMBL1745002

SCHEMBL1745002

C=CCc1cccc2c3c(ccc12)-c1ccccc1CN3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
CYP2C19 P33261 1/20 0.33
AKR1B1 P15121 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1745000 0.73 CA12 (0.33) GABRA1GABRB2CA12CA9ADRA1D
SCHEMBL5831594 0.71 GABRA1 (0.56) GABRA1GABRB2LMNAHTTKDM4E
SCHEMBL31619949 0.71 GABRA1 (0.56) GABRA1GABRB2LMNAHTTKDM4E
SCHEMBL458515 0.70 CA12 (0.44) CA12CA9LMNAHTTKDM4E
SCHEMBL16487340 0.67 GABRA1 (0.46) GABRA1GABRB2LMNAKDM4ECYP1A2
SCHEMBL30083977 0.67 GABRA1 (0.46) GABRA1GABRB2LMNAKDM4ECYP1A2
SCHEMBL5831736 0.67 GABRA1 (0.45) GABRA1GABRB2LMNAHTTKDM4E
SCHEMBL252161 0.66 PNMT (0.62) GABRA1GABRB2ADRA1DADRA1AADRA1B
SCHEMBL1147979 0.66 HPRT1 (0.52) GABRA1GABRB2LMNACYP1A2CYP2D6
SCHEMBL30083974 0.66 HPRT1 (0.52) GABRA1GABRB2LMNACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2387564-A1 BENZO ÝC¨PHENANTHRIDINES AS ANTIMICROBIAL AGENTS Rutgers, The State University of New Jersey (US) 2011-11-23 EP disclosed
US-8037884-B2 Modular system for patient positioning during medical procedures ALLEN MEDICAL SYSTEMS, INC. (US) 2011-10-18 US disclosed
WO-2010083436-A1 BENZO [C] PHENANTHRIDINES AS ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2010-07-22 WO disclosed