Piperidine

Piperidine

SCHEMBL17460237

C1CCNCC1.O=S1(=O)CCN(c2cccc(N3CCN(c4ccccc4)CC3)c2)CC1

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 7/20 0.54
ADRB1 P08588 3/20 0.49
HTR3E A5X5Y0 2/20 0.49
HTR3B O95264 2/20 0.49
HTR3A P46098 2/20 0.49
HTR3D Q70Z44 2/20 0.49
HTR3C Q8WXA8 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
HTR1A P08908 2/20 0.48
HTR7 P34969 2/20 0.48
HTR6 P50406 3/20 0.46
CYP2D6 P10635 3/20 0.45
HTR2C P28335 2/20 0.45
TP53 P04637 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
THRB P10828 1/20 0.45
CYP2C9 P11712 1/20 0.45
HTR2A P28223 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19281815 0.88 FAAH (0.65) FAAHKDM4EUSP2ALDH1A1TSHR
Piperidine SCHEMBL17460236 0.86 ADRB1 (0.49) FAAHADRB1HTR3EHTR3BHTR3A
SCHEMBL2456271 0.79 KDM4E (0.63) FAAHADRB1HTR3EHTR3BHTR3A
Piperidine SCHEMBL27934131 0.76 HTR3E (0.69) ADRB1HTR3EHTR3BHTR3AHTR3D
Pyrrolidine SCHEMBL28859475 0.76 HTR3E (0.69) ADRB1HTR3EHTR3BHTR3AHTR3D
Phenylpiperazine SCHEMBL3559958 0.76 ADRB1 (0.83) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL21963816 0.75 KDM4E (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL10510808 0.74 KDM4E (0.58) ADRB1HTR3EHTR3BHTR3AHTR3D
Pyrrolidine SCHEMBL12503448 0.74 HTR3E (0.72) ADRB1HTR3EHTR3BHTR3AHTR3D
Water SCHEMBL10512053 0.73 KDM4E (0.56) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014975-A2 UREA/CARBAMATES FAAH MAGL OR DUAL FAAH/MAGL INHIBITORS AND USES THEREOF NORTHEASTERN UNIVERSITY (US) 2016-01-28 WO disclosed