SCHEMBL17461544

SCHEMBL17461544

N=Cc1c(Nc2ccc(F)cc2)ccnc1CO

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 1/20 0.38
MAPT P10636 3/20 0.38
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
ALOX12 P18054 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
GAK O14976 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
KCNH2 Q12809 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
AURKA O14965 2/20 0.34
AURKB Q96GD4 2/20 0.34
KCNH3 Q9ULD8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17461535 0.75 MAPT (0.41) MAPK10MAPTPTGS1PTGS2RAB9A
SCHEMBL13393500 0.70 SMN1; SMN2 (0.32)
SCHEMBL17461539 0.66 RAB9A (0.52) MAPTPTGS1PTGS2RAB9AMEN1
SCHEMBL15673390 0.64 ERBB2 (0.66) MAPTGAKHTTERBB2CCNC
SCHEMBL17461534 0.64 PTGS1 (0.46) MAPTPTGS1PTGS2RAB9AMEN1
SCHEMBL24283166 0.61 MAPK10 (0.37) MAPK10MAPTPTGS1PTGS2RAB9A
SCHEMBL5473183 0.60 KMT2A (0.51) MAPTPTGS1RAB9AMEN1NPC1
SCHEMBL858107 0.60 TTBK1 (0.51) MAPK10MAPTRAB9AMEN1NPC1
SCHEMBL9402356 0.60 DHODH (0.57) MAPTRAB9ANPC1LMNAALOX12
SCHEMBL24003993 0.60 GAK (0.60) MAPTRAB9AMEN1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-B1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed