SCHEMBL17461534

SCHEMBL17461534

N=Cc1c(Br)cncc1Nc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 8/20 0.46
PTGS2 P35354 7/20 0.46
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
KCNH2 Q12809 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
SOS1 Q07889 1/20 0.36
MAPT P10636 2/20 0.34
BPTF Q12830 1/20 0.34
MEN1 O00255 1/20 0.33
PRKD3 O94806 1/20 0.33
EGFR P00533 1/20 0.33
PRKCG P05129 1/20 0.33
PRKCB P05771 1/20 0.33
SRC P12931 1/20 0.33
PRKCA P17252 1/20 0.33
PRKCH P24723 1/20 0.33
PRKCI P41743 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23912335 0.72 AOC1 (0.37)
SCHEMBL24283166 0.70 MAPK10 (0.37) PTGS1PTGS2ALDH1A1HTTRAB9A
SCHEMBL17461539 0.69 RAB9A (0.52) PTGS1PTGS2ALDH1A1HTTRAB9A
SCHEMBL567599 0.69 GAA (0.44) ALDH1A1HTTRAB9AKCNH2MAPT
SCHEMBL13393519 0.68 APP (0.33) PTGS1PTGS2
SCHEMBL23904233 0.67 MAPT (0.36) KCNH2SCN5ASCN9ASOS1MAPT
SCHEMBL20036833 0.66 MAPT (0.41) ALDH1A1HTTRAB9ASOS1MAPT
SCHEMBL17461544 0.64 MAPK10 (0.38) PTGS1PTGS2ALDH1A1HTTRAB9A
SCHEMBL17461535 0.64 MAPT (0.41) PTGS1PTGS2ALDH1A1HTTRAB9A
SCHEMBL30494419 0.64 CHRNB4 (0.48) PTGS1PTGS2ALDH1A1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-B1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed