SCHEMBL17469662

SCHEMBL17469662

CCCCNC(=N)c1ccc(NNc2c(N)ncc3ccc(Br)cc23)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.40
FLT3 P36888 1/20 0.40
NTRK3 Q16288 1/20 0.40
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RECQL P46063 1/20 0.31
EGFR P00533 1/20 0.31
KDR P35968 1/20 0.31
F2 P00734 1/20 0.31
EPHX2 P34913 1/20 0.31
AGPAT2 O15120 4/20 0.30
HDAC3 O15379 2/20 0.30
HDAC1 Q13547 2/20 0.30
HDAC2 Q92769 2/20 0.30
HDAC10 Q969S8 2/20 0.30
HDAC11 Q96DB2 2/20 0.30
HDAC8 Q9BY41 2/20 0.30
HDAC6 Q9UBN7 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17469641 0.85 KIT (0.47) KITFLT3NTRK3RAB9AF2
SCHEMBL17469656 0.82 KIT (0.43) KITFLT3NTRK3LMNASMN1; SMN2
SCHEMBL17469639 0.80 KIT (0.67) KITFLT3NTRK3NPC1RAB9A
SCHEMBL17469875 0.72 FLT3 (0.41) KITFLT3NTRK3EGFRF2
SCHEMBL21153064 0.71 KIT (0.56) KITFLT3NTRK3NPC1RAB9A
SCHEMBL17469797 0.69 CCNC (0.45)
SCHEMBL17469778 0.69 KIT (0.70) KITFLT3NTRK3NPC1RAB9A
SCHEMBL17469845 0.67 PRSS1 (0.42) LMNASMN1; SMN2EGFRKDRF2
SCHEMBL26485348 0.66 HDAC1 (0.43) LMNASMN1; SMN2F2HDAC1HDAC2
SCHEMBL31249942 0.66 HDAC3 (0.55) NPC1RAB9ALMNAHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014674-A1 LINKED DIARYL COMPOUNDS WITH ANTICANCER PROPERTIES AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2016-01-28 WO disclosed