SCHEMBL17477186

SCHEMBL17477186

CC1CN(C(=O)Oc2ccc(N)nc2)CCN1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 6/20 0.42
SCN10A Q9Y5Y9 2/20 0.42
HRH4 Q9H3N8 1/20 0.39
LIPE Q05469 3/20 0.39
TP53 P04637 1/20 0.39
MDM2 Q00987 1/20 0.39
ATR Q13535 1/20 0.38
GAA P10253 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
HDAC1 Q13547 1/20 0.38
REN P00797 1/20 0.38
PRKCQ Q04759 2/20 0.36
TRPC6 Q9Y210 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19066133 0.85 ALDH1A1 (0.46) LIPEGAAALDH1A1POLB
SCHEMBL17477123 0.83 HDAC1 (0.41) SCN9ASCN10AHRH4TP53MDM2
SCHEMBL4336868 0.80 GAA (0.60) HRH4TP53GAAALDH1A1REN
SCHEMBL25313933 0.78 ALDH1A1 (0.59) LIPEGAAALDH1A1POLB
SCHEMBL22635853 0.77 L3MBTL1 (0.47) SCN9AGAAALDH1A1POLB
SCHEMBL19066192 0.76 ALDH1A1 (0.67) LIPEGAAALDH1A1POLB
SCHEMBL4629620 0.75 HRH4 (0.40) SCN9ASCN10AHRH4TP53MDM2
SCHEMBL18191790 0.73 DPP4 (0.41) TRPC6
SCHEMBL28384237 0.73 HRH4 (0.39) SCN9ASCN10AHRH4TP53MDM2
SCHEMBL31112011 0.73 MLNR (0.50) HRH4GAAALDH1A1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015605-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed