SCHEMBL17481990

SCHEMBL17481990

Cc1ccc(C(=O)CCl)c2c1NC(=O)CO2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
ADRB1 P08588 10/20 0.37
ADRB2 P07550 7/20 0.37
DRD2 P14416 4/20 0.36
DRD4 P21917 4/20 0.36
DRD3 P35462 4/20 0.36
NR3C2 P08235 1/20 0.35
GAA P10253 1/20 0.34
HTR2A P28223 1/20 0.34
SMYD3 Q9H7B4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17481989 0.83 DRD2 (0.39) ALDH1A1ADRB1ADRB2DRD2DRD4
SCHEMBL8211174 0.83 DRD2 (0.39) ALDH1A1ADRB1ADRB2DRD2DRD4
SCHEMBL17481987 0.80 DRD2 (0.33) ALDH1A1MAPTADRB1ADRB2DRD2
SCHEMBL17484547 0.78 ADRB2 (0.39) ALDH1A1MAPTADRB1ADRB2DRD2
SCHEMBL11912374 0.77 DRD2 (0.42) ALDH1A1ADRB1ADRB2DRD2DRD4
SCHEMBL1559916 0.75 ADRB2 (0.39) ALDH1A1MAPTADRB1ADRB2DRD2
SCHEMBL17476304 0.75 SMYD3 (0.56) ALDH1A1MAPTDRD2GAASMYD3
SCHEMBL6428975 0.72 DRD2 (0.42) ALDH1A1ADRB1ADRB2DRD2DRD4
SCHEMBL8523943 0.71 ALDH1A1 (0.34) ALDH1A1MAPT
SCHEMBL9909524 0.69 DRD2 (0.58) ADRB1ADRB2DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9598381-B2 SMYD2 inhibitors ABBVIE INC. (US) 2017-03-21 US disclosed
US-20160031838-A1 SMYD2 INHIBITORS ABBVIE INC. 2016-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160031838-A1 SMYD2 INHIBITORS SMYD2, SMYD3, NSD1 ALDH1A1 3870/4885MAPT 2177/4885ADRB1 4623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.