SCHEMBL1748230

SCHEMBL1748230

N#Cc1ccc2sc(Cl)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.48
APP P05067 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
IDO1 P14902 1/20 0.40
DYRK1A Q13627 1/20 0.39
MIF P14174 1/20 0.39
KMT2A Q03164 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP2A6 P11509 1/20 0.37
PSMB8 P28062 2/20 0.37
PSMB5 P28074 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1032990 0.86 APP (0.55) APPSMN1; SMN2NPSR1DYRK1AMIF
SCHEMBL507628 0.80 PPARA (0.49) PPARAAPPDYRK1ACYP2A6KDM4E
SCHEMBL1997208 0.79 PPARA (0.48) PPARAAPPDYRK1ACYP2A6KDM4E
SCHEMBL7380470 0.79 SMN1; SMN2 (0.52) PPARAAPPSMN1; SMN2DYRK1AKMT2A
SCHEMBL12298168 0.79 PPARA (0.48) PPARAAPPDYRK1ACYP2A6KDM4E
SCHEMBL30602948 0.79 PPARA (0.48) PPARAAPPDYRK1ACYP2A6KDM4E
SCHEMBL9808445 0.79 CYP3A4 (0.51) PPARAAPPSMN1; SMN2NPC1RAB9A
SCHEMBL780242 0.77 SMN1; SMN2 (0.61) PPARASMN1; SMN2NPSR1LOXL2IDO1
SCHEMBL24963247 0.75 LOXL2 (0.59) PPARAAPPLOXL2DYRK1ANPC1
SCHEMBL1747932 0.75 PPARA (0.61) PPARAAPPSMN1; SMN2NPSR1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024117179-A1 KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF ALIVEXIS, INC. (JP) 2024-06-06 WO disclosed
EP-3397629-B1 METALLOENZYME INHIBITOR COMPOUNDS NQP 1598 LTD (KY) 2023-04-19 EP disclosed
EP-3397629-B1 METALLOENZYME INHIBITOR COMPOUNDS NQP 1598 LTD (KY) 2023-04-19 EP disclosed
EP-4141002-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS Incyte Corporation (US) 2023-03-01 EP disclosed
US-11572366-B2 Heterocyclic compounds as immunomodulators INCYTE CORPORATION (US) 2023-02-07 US disclosed
CN-109641885-B Heterocyclic compounds as immunomodulators 因赛特公司 2022-09-30 CN disclosed
EP-3377488-B1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORP (US) 2022-08-10 EP disclosed
US-20210221819-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2021-07-22 US disclosed
US-10464922-B2 Metalloenzyme inhibitor compounds NQP 1598, LTD. (US) 2019-11-05 US disclosed
CN-109641885-A Heterocyclic compound as immunomodulator 因赛特公司 2019-04-16 CN disclosed
US-20030171399-A1 Quinolinyl and benzothiazolyl modulators TULARIK INC. 2003-09-11 US disclosed
CN-1438998-A Quinolinyl and benzothiazolyl PPAR-gamma modulators TULARIK INC (US) 2003-08-27 CN disclosed
US-6583157-B2 Peroxisome proliferator-activated receptors antagonists; antiinflammatory agents and treating metabolic disorders TULARIK INC. 2003-06-24 US disclosed
EP-1296967-A1 QUINOLINYL AND BENZOTHIAZOLYL PPAR-GAMMA MODULATORS Tularik Inc. (US) 2003-04-02 EP disclosed
US-20020169185-A1 QUINOLINYL AND BENZOTHIAZOLYL MODULATORS AMGEN INC. 2002-11-14 US disclosed
WO-2002000633-A1 QUINOLINYL AND BENZOTHIAZOLYL PPAR-GAMMA MODULATORS TULARIK INC. (US) 2002-01-03 WO disclosed
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0129506-B1 HETEROCYCLICALLY SUBSTITUTED THIO(CYCLO)ALKANE POLYCARBOXYLIC ACIDS CIBA-GEIGY AG (CH) 1991-03-06 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210221819-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS CD74, IL2, ICOS PPARA 639/4885APP 4745/4885SMN1; SMN2 4119/4885
US-10464922-B2 Metalloenzyme inhibitor compounds MMEL1, GPX1, MPO PPARA 3103/4885APP 1437/4885SMN1; SMN2 1142/4885
US-20030171399-A1 Quinolinyl and benzothiazolyl modulators PPARA, PPARG, PPARD PPARA 1/4885APP 3233/4885SMN1; SMN2 4885/4885
US-20020169185-A1 QUINOLINYL AND BENZOTHIAZOLYL MODULATORS PPARA, PPARG, PPARD PPARA 1/4885APP 3233/4885SMN1; SMN2 4885/4885
US-11572366-B2 Heterocyclic compounds as immunomodulators CD74, IL2, ICOS PPARA 639/4885APP 4745/4885SMN1; SMN2 4119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.