SCHEMBL1748238

SCHEMBL1748238

Cc1ccc2nc(Nc3ccc(-c4ccc(C(=O)[C@@H]5CCC[C@@]5(C)C(=O)O)cc4)cc3F)oc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.42
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
ATM Q13315 1/20 0.36
GALK1 P51570 8/20 0.35
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
MAP4K4 O95819 1/20 0.35
ABL1 P00519 1/20 0.35
LCK P06239 1/20 0.35
FYN P06241 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL2311135 0.84 DGAT1 (0.44) DGAT1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL1748140 0.83 DGAT1 (0.58) DGAT1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL1748237 0.80 DGAT1 (0.49) DGAT1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL12315617 0.79 DGAT1 (0.46) DGAT1SMN1; SMN2KDM4EALDH1A1MAPT
Bicarbonate SCHEMBL2359226 0.77 DGAT1 (0.42) DGAT1MAPTNPC1RAB9ADYRK3
SCHEMBL2308158 0.76 DGAT1 (0.56) DGAT1MAPTNPC1RAB9ADYRK3
SCHEMBL1748065 0.76 DGAT1 (0.41) DGAT1SMN1; SMN2KDM4EMAPTHSD17B10
SCHEMBL2309580 0.76 DGAT1 (0.41) DGAT1KDM4EHSD17B10
Bicarbonate SCHEMBL2314871 0.75 DGAT1 (0.51) DGAT1SMN1; SMN2GALK1CSF1RHDAC6
SCHEMBL2309693 0.74 DGAT1 (0.67) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8013166-B2 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER HEALTHCARE LLC (US) 2011-09-06 US disclosed
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP disclosed