SCHEMBL17486170

SCHEMBL17486170

Cc1cnc(-c2ccc3c(c2)C2CCC3C2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
PDK2 Q15119 2/20 0.36
PDK4 Q16654 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
DGAT1 O75907 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CNR2 P34972 1/20 0.32
RARG P13631 2/20 0.31
RARB P10826 1/20 0.31
NOTUM Q6P988 1/20 0.31
JAK3 P52333 1/20 0.31
DHODH Q02127 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486224 0.84 KDM1A (0.35) SIGMAR1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL19295089 0.78 LPL (0.37) DGAT1
SCHEMBL17486228 0.76 ALDH1A1 (0.34) SIGMAR1CHRNB2CHRNA4CNR2RARG
SCHEMBL17486185 0.76 CYP11B1 (0.35) SIGMAR1CYP11B1CYP11B2
SCHEMBL17485979 0.75 IKBKB (0.36) SIGMAR1PDK2PDK4CNR2RARG
SCHEMBL20805515 0.75 CYP11B1 (0.35) CYP11B1CYP11B2
SCHEMBL24602339 0.72 RPS6KA3 (0.45) CYP11B1CYP11B2DHODH
SCHEMBL17485972 0.72 SIGMAR1 (0.33) SIGMAR1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17486126 0.71 KDM1A (0.33) SIGMAR1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17486157 0.71 PTGDR2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed