SCHEMBL17486228

SCHEMBL17486228

Cc1cc(Br)cnc1-c1ccc2c(c1)C1CCC2C1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
DHODH Q02127 2/20 0.32
CNR2 P34972 1/20 0.32
NOTUM Q6P988 2/20 0.31
RARG P13631 2/20 0.30
RARB P10826 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486224 0.86 KDM1A (0.35) ALDH1A1MAPTMAPK1HTTSMN1; SMN2
SCHEMBL17486287 0.80 CHRNA1 (0.34) ALDH1A1MAPTCHRNB2CHRNA4JAK3
SCHEMBL17486170 0.76 SIGMAR1 (0.39) SIGMAR1CHRNB2CHRNA4DHODHCNR2
SCHEMBL19295072 0.75 HSD17B1 (0.34) MAPK1SMN1; SMN2
SCHEMBL19295168 0.75 PPARA (0.33) MAPTSMN1; SMN2
SCHEMBL19295078 0.75 IKBKB (0.35) CNR2RARGRARB
SCHEMBL17485995 0.75 GRM5 (0.34) SIGMAR1CHRNB2CHRNA4NOTUM
SCHEMBL17486052 0.74 DHODH (0.35) SIGMAR1DHODH
SCHEMBL17486043 0.74 CAMKK2 (0.36) SIGMAR1JAK3
SCHEMBL10472664 0.73 SMN1; SMN2 (0.47) ALDH1A1MAPTMAPK1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170250353-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 ALDH1A1 3721/4885MAPT 1084/4885MAPK1 4229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.