SCHEMBL17486273

SCHEMBL17486273

CC12CCC(C)(O1)c1cc(-c3ccc(Br)cn3)ccc12

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
NFKB1 P19838 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.35
BACE1 P56817 2/20 0.34
CA2 P00918 1/20 0.33
CYP1A1 P04798 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP1B1 Q16678 1/20 0.32
ALOX5AP P20292 1/20 0.30
RARG P13631 1/20 0.30
PTPN1 P18031 1/20 0.30
PTPN6 P29350 1/20 0.30
CDC25A P30304 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16812192 0.82 HSD17B1 (0.41) NPC1RAB9ABACE1RARG
SCHEMBL17486216 0.81 MAPK1 (0.37) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL18015246 0.81 RARA (0.44) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL20007152 0.81 NPC1 (0.37) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL17486214 0.79 BACE1 (0.32) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL17486213 0.78 NPC1 (0.35) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL15614853 0.78 KDM1A (0.36) BACE1
SCHEMBL18015415 0.78 NPC1 (0.37) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL19295085 0.78 DGAT1 (0.49) BACE1
SCHEMBL19295154 0.77 MEN1 (0.38) L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170250353-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 NPC1 3516/4885NFKB1 1929/4885MAPK1 4229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.