SCHEMBL17486348

SCHEMBL17486348

CCc1cc2c(cc1-c1ccc(-c3nc(-c4ccccc4)nc(-c4ccccc4)n3)cn1)C(C)(C)C(C)(C)C2(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.35
KMT2A Q03164 6/20 0.35
ALDH1A1 P00352 5/20 0.35
MAPT P10636 5/20 0.35
HPGD P15428 5/20 0.35
KDM4E B2RXH2 3/20 0.35
ADORA2A P29274 3/20 0.33
ADORA1 P30542 3/20 0.33
ADORA3 P0DMS8 2/20 0.33
ADORA2B P29275 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP2C19 P33261 1/20 0.32
NTSR1 P30989 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486208 0.93 MEN1 (0.34) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL17486349 0.93 KDM4E (0.37) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL17486350 0.90 CYP2A6 (0.39) MAPTNPC1RAB9ASMN1; SMN2CYP2C19
SCHEMBL17486202 0.87 RARG (0.35) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL17486212 0.87 MEN1 (0.34) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL17486251 0.85
SCHEMBL17486354 0.84 CYP1A2 (0.41) NPC1ALOX5APFEN1
SCHEMBL17486352 0.84 DGAT1 (0.32) MAPT
SCHEMBL17486353 0.83 SMN1; SMN2 (0.35) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL17486227 0.82 HSD17B1 (0.41) MEN1KMT2AALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed