SCHEMBL174937

SCHEMBL174937

C=CC(=O)NCNC(=O)c1ccccc1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
TSHR P16473 2/20 0.48
MAPK1 P28482 1/20 0.48
CYP1A2 P05177 1/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.40
TGM2 P21980 5/20 0.38
MAPT P10636 2/20 0.37
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
TP53 P04637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
HTT P42858 1/20 0.35
TRIM24 O15164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5459625 0.81 GAA (0.42) TDP1TSHRCYP1A2HPGDGAA
SCHEMBL3093204 0.79 CYP1A2 (0.42) TDP1TSHRCYP1A2HPGDMAPT
SCHEMBL3285344 0.79 ALDH1A1 (0.61) ALDH1A1TDP1TSHRMAPK1GAA
SCHEMBL10279067 0.77 LMNA (0.43) ALDH1A1TDP1TSHRCYP1A2HPGD
SCHEMBL27521277 0.76 HTT (0.45) TDP1TSHRCYP1A2HPGDMEN1
SCHEMBL16157270 0.76 KMT2A (0.41) TDP1TSHRCYP1A2HPGDMEN1
SCHEMBL10117106 0.76 KMT2A (0.49) ALDH1A1TDP1TSHRHPGDCA1
SCHEMBL15728763 0.76 KEAP1 (0.53) TDP1GAAMAPTMEN1LMNA
SCHEMBL6609811 0.74 ALDH1A1 (0.51) ALDH1A1TSHRHPGDMAPTMEN1
SCHEMBL27503407 0.74 HTT (0.50) ALDH1A1TSHRHPGDMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2795406-B1 ALCOHOL-SOLUBLE HOLE TRANSPORT MATERIALS FOR ORGANIC PHOTOCONDUCTOR COATINGS HEWLETT PACKARD DEVELOPMENT CO LP (US) 2017-02-08 EP disclosed
US-9482970-B2 Organic photoconductors having protective coatings with nanoparticles HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2016-11-01 US disclosed
EP-2831674-B1 ORGANIC PHOTOCONDUCTORS HAVING PROTECTIVE COATINGS WITH NANOPARTICLES HEWLETT PACKARD DEVELOPMENT CO (US) 2016-03-30 EP disclosed
US-9235147-B2 Alcohol-soluble hole transport materials for organic photoconductor coatings HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2016-01-12 US disclosed
US-9188884-B2 Charge transport layer for organic photoconductors HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2015-11-17 US disclosed
EP-2611872-B1 INKJET PRINTING FLUID EASTMAN KODAK CO (US) 2015-07-08 EP disclosed
EP-2831674-A1 ORGANIC PHOTOCONDUCTORS HAVING PROTECTIVE COATINGS WITH NANOPARTICLES Hewlett-Packard Development Company, L.P. (US) 2015-02-04 EP disclosed
US-20140349227-A1 ORGANIC PHOTOCONDUCTORS HAVING PROTECTIVE COATINGS WITH NANOPARTICLES HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. 2014-11-27 US disclosed
US-20140322638-A1 ALCOHOL-SOLUBLE HOLE TRANSPORT MATERIALS FOR ORGANIC PHOTOCONDUCTOR COATINGS HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2014-10-30 US disclosed
EP-2794785-A1 INKJET INK COMPOSITION Eastman Kodak Company (US) 2014-10-29 EP disclosed
US-5958661-A HAVING GREEN LIGHT SENSITIVE MAGENTA DYE FORMING LAYER CONTAINING PYRAZOLOAZOLE DYE FORMING COUPLER EASTMAN KODAK COMPANY (US) 1999-09-28 US disclosed
EP-0727704-B1 Method for forming photographic dispersions comprising loaded latex polymers EASTMAN KODAK CO (US) 1999-04-21 EP disclosed
EP-0727705-B1 Photographic print material EASTMAN KODAK CO (US) 1998-12-09 EP disclosed
EP-0727703-B1 Method for preparing photographic elements comprising loaded latex compositions EASTMAN KODAK CO (US) 1998-11-11 EP disclosed
US-5594047-A Method for forming photographic dispersions comprising loaded latex polymers EASTMAN KODAK COMPANY (US) 1997-01-14 US disclosed
US-5582960-A COLOR PHOTOGRAPHIC IMAGE DISPLAY MATERIAL COMPRISING YELLOW DYE-FORMING BLUE LIGHT SENSITIVE SILVER HALIDE EMULSION LAYER INCLUDING SILVER CHLORIDE SPECTRALLY SENSITIZED WITH SPECIFIED DYE, SPECIFIED COUPLER, WATER INSOLUBLE POLYMER EASTMAN KODAK COMPANY (US) 1996-12-10 US disclosed
US-5558980-A FORMING A PHOTOGRAPHIC FILM FORMING LAYERS OF COLLOIDS, SURFACTANTS AND LATEX EASTMAN KODAK COMPANY (US) 1996-09-24 US disclosed
EP-0727703-A1 Method for preparing photographic elements comprising loaded latex compositions EASTMAN KODAK COMPANY (US) 1996-08-21 EP disclosed
EP-0727705-A1 Photographic print material EASTMAN KODAK COMPANY (US) 1996-08-21 EP disclosed
EP-0727704-A1 Method for forming photographic dispersions comprising loaded latex polymers EASTMAN KODAK COMPANY (US) 1996-08-21 EP disclosed