SCHEMBL17508314

SCHEMBL17508314

O=Cc1ccc(Cc2cc(F)c(F)c(F)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
KIF11 P52732 1/20 0.40
ALDH1A1 P00352 7/20 0.38
CYP2A6 P11509 3/20 0.37
HSD17B10 Q99714 1/20 0.37
ALDH5A1 P51649 1/20 0.37
ABAT P80404 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ALDH3A1 P30838 1/20 0.35
ALDH1A3 P47895 1/20 0.35
PTGER4 P35408 1/20 0.35
TUBB1 Q9H4B7 1/20 0.33
TYR P14679 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17508169 0.84 CYP17A1 (0.44) KMT2AKIF11ALDH1A1CYP2A6HSD17B10
SCHEMBL3976211 0.80 CYP2A6 (0.52) KMT2AALDH1A1CYP2A6HSD17B10ALDH5A1
SCHEMBL9607165 0.79 KMT2A (0.61) KMT2AALDH1A1CYP2A6HSD17B10ALDH5A1
SCHEMBL16105658 0.78 CES2 (0.39) MAOB
SCHEMBL12889505 0.75 CYP1A2 (0.41) ALDH1A1CYP2A6MAPTMAOB
SCHEMBL16037967 0.75 KIF11 (0.59) KIF11ALDH1A1CYP2A6HSD17B10ALDH5A1
SCHEMBL17508154 0.75 KMT2A (0.41) KMT2AKIF11ALDH1A1CYP2A6HSD17B10
SCHEMBL18351321 0.74 CYP17A1 (0.40) ALDH1A1MAOAMAOB
SCHEMBL7239271 0.74 LTA4H (0.35) TUBB1
SCHEMBL17508269 0.73 CYP2A6 (0.54) KMT2AALDH1A1CYP2A6HSD17B10ALDH5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed