SCHEMBL17508994

SCHEMBL17508994

OB(Cc1ccccc1)OOC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
GRIN2B Q13224 1/20 0.33
LIPE Q05469 1/20 0.33
ARG2 P78540 1/20 0.32
TSHR P16473 2/20 0.32
TRPV6 Q9H1D0 1/20 0.32
SLC6A2 P23975 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
PLA2G1B P04054 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ATG4B Q9Y4P1 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
FAAH O00519 3/20 0.31
PDK2 Q15119 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23535576 0.75 LIPE (0.39) CA1CA2LIPEARG2TSHR
SCHEMBL874879 0.71 TRPV6 (0.42) CES1CA1CA2TSHRTRPV6
SCHEMBL3900187 0.70 CA1 (0.41) CA1CA2LIPEARG2TSHR
SCHEMBL1356582 0.70 CA1 (0.41) CES1CA1CA2LIPEARG2
SCHEMBL670441 0.69 LIPE (0.35) CA1CA2LIPEARG2TSHR
SCHEMBL17508991 0.68 EPHX2 (0.38) CES1GRIN2BTSHR
SCHEMBL3887273 0.68 TSHR (0.46) CA1CA2LIPEARG2TSHR
SCHEMBL28070120 0.68 CA1 (0.34) CA1CA2TSHRTRPV6PDK2
SCHEMBL5952624 0.68 TRPA1 (0.39) CA1CA2LIPETSHRSLC6A2
SCHEMBL25377641 0.66 CA1 (0.46) CA1CA2LIPEARG2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180340-A1 PYRIDO[2,3-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES Hydra Biosciences, Inc. (US) 2017-06-21 EP disclosed
WO-2016023830-A1 PYRIDO[2,3-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES HYDRA BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed