SCHEMBL175193

SCHEMBL175193

COC(=O)CCc1ccc(C(=O)c2sc(N)nc2-c2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
HSD17B10 Q99714 1/20 0.52
LMNA P02545 4/20 0.50
NPSR1 Q6W5P4 4/20 0.50
HTT P42858 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
POLB P06746 2/20 0.50
MAPT P10636 2/20 0.50
ADORA1 P30542 5/20 0.49
ADORA3 P0DMS8 8/20 0.48
ADORA2B P29275 2/20 0.47
ADORA2A P29274 1/20 0.45
GAA P10253 2/20 0.44
PKM P14618 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
RORC P51449 1/20 0.43
RORB Q92753 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4267596 0.83 ALDH1A1 (0.55) ALDH1A1HSD17B10LMNANPSR1HTT
SCHEMBL176165 0.83 ALDH1A1 (0.55) ALDH1A1HSD17B10LMNANPSR1HTT
SCHEMBL175366 0.81 ALDH1A1 (0.53) ALDH1A1HSD17B10LMNANPSR1HTT
SCHEMBL165773 0.79 ADORA3 (0.61) ALDH1A1HSD17B10LMNANPSR1HTT
SCHEMBL5397061 0.79 CYP1A2 (0.60) ALDH1A1HSD17B10LMNAHTTSMN1; SMN2
SCHEMBL257616 0.76 ADORA3 (0.64) ALDH1A1HSD17B10LMNANPSR1SMN1; SMN2
SCHEMBL11629832 0.75 SRD5A2 (0.56) ALDH1A1HTTSMN1; SMN2MAPTKMT2A
SCHEMBL27653923 0.75 ALDH1A1 (0.64) ALDH1A1HSD17B10NPSR1HTTSMN1; SMN2
SCHEMBL174332 0.75 SMN1; SMN2 (0.54) ALDH1A1HSD17B10LMNANPSR1HTT
SCHEMBL19669120 0.74 ALDH1A1 (0.72) ALDH1A1HSD17B10SMN1; SMN2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed