SCHEMBL174332

SCHEMBL174332

COC(=O)c1cccc(-c2nc(N)sc2C(=O)c2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
LMNA P02545 3/20 0.54
NPSR1 Q6W5P4 3/20 0.54
HTT P42858 2/20 0.54
MAPT P10636 1/20 0.54
RORB Q92753 7/20 0.54
ALDH1A1 P00352 4/20 0.53
HSD17B10 Q99714 2/20 0.53
POLB P06746 1/20 0.51
KDM4E B2RXH2 1/20 0.50
HPGD P15428 1/20 0.50
ADORA3 P0DMS8 4/20 0.49
ADORA1 P30542 2/20 0.49
ADORA2B P29275 2/20 0.48
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165773 0.83 ADORA3 (0.61) SMN1; SMN2LMNANPSR1HTTMAPT
SCHEMBL257432 0.81 RORB (0.74) LMNANPSR1RORBALDH1A1HSD17B10
SCHEMBL19669120 0.81 ALDH1A1 (0.72) SMN1; SMN2MAPTALDH1A1HSD17B10POLB
SCHEMBL175512 0.79 RORB (0.54) RORBALDH1A1HSD17B10ADORA3ADORA1
SCHEMBL169403 0.78 RORC (0.58) SMN1; SMN2LMNANPSR1HTTMAPT
SCHEMBL10092883 0.77 RORB (0.67) RORBALDH1A1HSD17B10ADORA3ADORA1
SCHEMBL27653923 0.76 ALDH1A1 (0.64) SMN1; SMN2NPSR1HTTMAPTRORB
SCHEMBL257615 0.75 RORB (0.72) RORBALDH1A1
SCHEMBL14364298 0.75 KDM4E (0.54) SMN1; SMN2LMNAMAPTALDH1A1HSD17B10
SCHEMBL175193 0.75 ALDH1A1 (0.52) SMN1; SMN2LMNANPSR1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed