SCHEMBL17523673

SCHEMBL17523673

NCCC(=C(c1ccccc1)c1ccccc1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.61
ESR1 P03372 11/20 0.55
CYP19A1 P11511 10/20 0.50
ESR2 Q92731 9/20 0.50
CYP3A4 P08684 2/20 0.50
ESRRB O95718 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2A6 P11509 1/20 0.45
CYP3A5 P20815 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17506008 0.84 PTGS2 (0.58) PTGS2ESR1CYP19A1ESR2CYP3A4
SCHEMBL17506000 0.82 CYP19A1 (0.78) ESR1CYP19A1ESR2CYP3A4CYP1A2
SCHEMBL9100272 0.81 PTGS2 (0.61) PTGS2ESR1CYP19A1ESR2ESRRB
SCHEMBL19182067 0.80 CYP19A1 (0.65) ESR1CYP19A1ESR2CYP3A4ESRRB
SCHEMBL17523634 0.80 CYP19A1 (0.65) ESR1CYP19A1ESR2CYP3A4ESRRB
SCHEMBL8615209 0.79 ESR1 (0.81) PTGS2ESR1CYP19A1ESR2
SCHEMBL7712232 0.79 PTGS2 (0.44) PTGS2ESR1CYP19A1ESR2CYP3A4
SCHEMBL11043479 0.77 PTGS2 (0.42) PTGS2ESR1CYP19A1ESR2CYP3A4
SCHEMBL9860588 0.77 PTGS2 (0.68) PTGS2ESR1ESR2ESRRB
SCHEMBL28108412 0.76 PTGS2 (1.00) PTGS2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170217914-A1 Novel Triarylethylene Compounds and Methods Using Same THE PENN STATE RESEARCH FOUNDATION 2017-08-03 US disclosed
US-20170217914-A1 Novel Triarylethylene Compounds and Methods Using Same THE PENN STATE RESEARCH FOUNDATION 2017-08-03 US disclosed
WO-2016022325-A1 NOVEL TRIARYLETHYLENE COMPOUNDS AND METHODS USING SAME THE PENN STATE RESEARCH FOUNDATION (US) 2016-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170217914-A1 Novel Triarylethylene Compounds and Methods Using Same CYP46A1, GSTA2, GSTA1 PTGS2 1024/4885ESR1 1247/4885CYP19A1 34/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.