SCHEMBL17524917

SCHEMBL17524917

C[Si](C)(C)CCOCN1C(=O)C2(CCN(c3ccc(N)cc3)CC2)c2cc(Br)cnc21

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.33
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524871 0.89 OPRM1 (0.33)
SCHEMBL21912465 0.87 DGAT1 (0.31) DGAT1
SCHEMBL17506487 0.85 NPC1 (0.34)
SCHEMBL17525045 0.85 EGLN1 (0.41) EGLN1
SCHEMBL15699637 0.85 CALCRL (0.31)
SCHEMBL17506429 0.80 GAA (0.37)
SCHEMBL15699763 0.79 NAMPT (0.37)
SCHEMBL17525046 0.77 OPRL1 (0.35) EGLN1
SCHEMBL722670 0.76 DGAT1 (0.33) DGAT1
SCHEMBL15882578 0.76 DGAT1 (0.32) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed