SCHEMBL17525955

SCHEMBL17525955

CO[C@H]1CCC2C3CCc4c(ccc(C#N)c4C)C3CC[C@@]21C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.47
MAPT P10636 5/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
ESR2 Q92731 4/20 0.47
MAPK1 P28482 3/20 0.47
LMNA P02545 3/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
G6PD P11413 1/20 0.47
PKM P14618 1/20 0.47
MPI P34949 1/20 0.47
CYP3A4 P08684 3/20 0.46
ALOX15 P16050 2/20 0.46
BRCA1 P38398 1/20 0.46
RECQL P46063 1/20 0.46
CYP19A1 P11511 2/20 0.44
TP53 P04637 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
PTPN11 Q06124 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17525951 0.88 CYP19A1 (0.53) ESR1MAPTMEN1KMT2AESR2
SCHEMBL17525983 0.80 MAPT (0.44) ESR1MAPTMEN1KMT2AESR2
SCHEMBL29470239 0.79 ESR1 (0.61) ESR1MAPTMEN1KMT2AESR2
SCHEMBL14048666 0.78 LMNA (0.56) ESR1MAPTMEN1KMT2AESR2
SCHEMBL13952052 0.77 STS (0.50) ESR1MAPTMEN1KMT2AESR2
SCHEMBL13951889 0.76 STS (0.69) ESR1MAPTESR2LMNACYP3A4
SCHEMBL14048673 0.76 SHBG (0.50) ESR1MAPTMEN1KMT2AESR2
SCHEMBL13952055 0.75 STS (0.61) ESR1MAPTESR2LMNACYP3A4
SCHEMBL14048668 0.73 STS (0.51) ESR1MAPTMEN1KMT2AESR2
SCHEMBL8508439 0.73 ESR1 (0.46) ESR1MAPTMEN1KMT2AESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2147014-B1 17ALPHA-SUBSTITUTED STEROIDS AS SYSTEMIC ANTIANDROGENS AND SELECTIVE ANDROGEN RECEPTOR MODULATORS ENDORECH INC (CA) 2016-02-17 EP disclosed