SCHEMBL17529970

SCHEMBL17529970

COc1cc(F)cc(C2CCN(C(=O)C(CC(C)C)NC(=O)CC#N)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 6/20 0.44
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
ADAMTS4 O75173 2/20 0.38
ADAMTS5 Q9UNA0 2/20 0.38
SMYD3 Q9H7B4 1/20 0.38
CTSL P07711 3/20 0.37
CTSK P43235 3/20 0.37
CTSS P25774 2/20 0.37
ACACB O00763 1/20 0.37
CCKBR P32239 1/20 0.36
CTSB P07858 2/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
ROCK2 O75116 1/20 0.35
PRKG1 Q13976 1/20 0.35
CACNA1B Q00975 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17530237 0.82 CTSS (0.52) CTSLCTSKCTSSCTSBROCK2
SCHEMBL17530381 0.81 CCR1 (0.62) CCR1CTSLCTSKCTSSCCKBR
SCHEMBL17530229 0.78 CTSL (0.50) CTSLCTSKCTSSCTSB
SCHEMBL17529981 0.75 CTSS (0.48) CTSLCTSKCTSSCTSB
SCHEMBL17530335 0.70 CTSS (0.55) CTSLCTSKCTSSCTSB
SCHEMBL19702755 0.69 ALDH1A1 (0.51) ALDH1A1
SCHEMBL17530252 0.69 CTSS (0.53) CTSLCTSKCTSSCTSBROCK2
SCHEMBL17529983 0.67 CTSS (0.57) CCR1CTSLCTSKCTSSCTSB
SCHEMBL17530018 0.67 CCR1 (0.42) CCR1CTSLCTSKCTSSACACB
SCHEMBL17530369 0.66 CTSL (0.59) CTSLCTSKCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027284-A2 PIPERIDINE UREAS AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed